SCHEMBL28825532

SCHEMBL28825532

[CH2]c1ccccc1-n1ccc(-c2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 2/20 0.44
GABRA1 P14867 1/20 0.44
HPGD P15428 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
LMNA P02545 2/20 0.44
IDO1 P14902 1/20 0.42
CAPN1 P07384 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CTSS P25774 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6697417 0.81 ALDH1A1 (0.66) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL19657972 0.75 ALDH1A1 (0.70) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL9383785 0.74 KDM4E (0.56) CYP1A2CYP3A4ALDH1A1KDM4EGABRA1
SCHEMBL13733242 0.74 ALDH1A1 (0.52) CYP1A2CYP3A4ALDH1A1KDM4EGABRA1
SCHEMBL98946 0.72 KDM4E (0.41) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL26253632 0.71 KDM4E (0.52) CYP1A2CYP3A4ALDH1A1KDM4EGABRA1
SCHEMBL12777946 0.70 ALDH1A1 (0.51) CYP1A2CYP3A4ALDH1A1KDM4EGABRA1
SCHEMBL2091831 0.69 RORC (0.50) ALDH1A1KDM4EHPGDIDO1MAOB
SCHEMBL2710665 0.68 ALDH1A1 (0.60) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL4723906 0.68 HDAC1 (0.51) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed