SCHEMBL13733889

SCHEMBL13733889

NC(=O)c1c(F)ccc(OCCc2nc(-c3ccc(C(F)(F)F)cc3)co2)c1F

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.40
S1PR3 Q99500 3/20 0.40
PARP1 P09874 1/20 0.35
SCN9A Q15858 8/20 0.35
IKBKB O14920 1/20 0.34
CASP1 P29466 1/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
CHEK2 O96017 1/20 0.33
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13732923 0.89 S1PR1 (0.37) S1PR1S1PR3PARP1SCN9A
SCHEMBL13731435 0.86 S1PR1 (0.39) S1PR1S1PR3PARP1IKBKBCASP1
SCHEMBL13733290 0.81 IKBKB (0.35) S1PR1SCN9AIKBKBPPARGPPARA
SCHEMBL13732543 0.81 SCN9A (0.35) S1PR1S1PR3PARP1SCN9AIKBKB
SCHEMBL13734892 0.81 IKBKB (0.35) S1PR1SCN9AIKBKBPPARGPPARA
SCHEMBL13732676 0.81 IKBKB (0.35) IKBKBCASP1PPARGPPARA
SCHEMBL203408 0.80 HSD17B1 (0.33) S1PR1S1PR3SCN9A
SCHEMBL2706695 0.79 MAPT (0.37) S1PR1S1PR3SCN9A
SCHEMBL17275080 0.79 HDAC3 (0.52)
SCHEMBL13732485 0.78 SCN9A (0.39) S1PR1S1PR3SCN9ACASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699557-A1 AROMATIC AMIDES AND USES THEREOF Biota Scientific Management Pty Ltd (AU) 2014-02-26 EP disclosed
WO-2012142671-A1 AROMATIC AMIDES AND USES THEREOF BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2012-10-26 WO disclosed