SCHEMBL137348

SCHEMBL137348

O=C(CCCCCCC(=O)Nc1ccccc1)Nc1ccccc1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 19/20 0.85
HDAC1 Q13547 19/20 0.85
HDAC11 Q96DB2 19/20 0.85
HDAC8 Q9BY41 19/20 0.85
HDAC6 Q9UBN7 19/20 0.85
HDAC5 Q9UQL6 19/20 0.85
HDAC7 Q8WUI4 18/20 0.85
HDAC9 Q9UKV0 18/20 0.85
HDAC3 O15379 18/20 0.85
HDAC2 Q92769 18/20 0.85
HDAC10 Q969S8 18/20 0.85
NCOR1 O75376 2/20 0.85
NCOR2 Q9Y618 2/20 0.85
KDM4E B2RXH2 1/20 0.85
BRD4 O60885 1/20 0.85
NR1I2 O75469 1/20 0.85
EGFR P00533 1/20 0.85
CYP3A4 P08684 1/20 0.85
LTA4H P09960 1/20 0.85
NR0B1 P51843 1/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665592 1.00 HDAC4 (0.85) HDAC4HDAC1HDAC11HDAC8HDAC6
SCHEMBL6669511 1.00 HDAC4 (0.85) HDAC4HDAC1HDAC11HDAC8HDAC6
SCHEMBL1065393 1.00 HDAC4 (0.85) HDAC4HDAC1HDAC11HDAC8HDAC6
SCHEMBL517309 0.98 HDAC4 (0.81) HDAC4HDAC1HDAC11HDAC8HDAC6
Hydroxyamine SCHEMBL1268824 0.96 HDAC6 (0.79) HDAC4HDAC1HDAC11HDAC8HDAC6
SCHEMBL1064861 0.94 HDAC4 (0.77) HDAC4HDAC1HDAC11HDAC8HDAC6
SCHEMBL312344 0.94 HDAC4 (0.77) HDAC4HDAC1HDAC11HDAC8HDAC6
SCHEMBL6296181 0.93 HDAC4 (0.75) HDAC4HDAC1HDAC11HDAC8HDAC6
SCHEMBL23055010 0.92 HDAC1 (1.00) HDAC4HDAC1HDAC11HDAC8HDAC6
SCHEMBL4403514 0.92 HDAC8 (0.74) HDAC4HDAC1HDAC11HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 901 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024014643-A1 METHOD FOR PRODUCING IMMUNOCYTES HAVING IMPROVED CYTOTOXICITY 주식회사 노보셀바이오 2024-01-18 WO claimed
WO-2023201270-A2 THERAPEUTIC APPLICATIONS OF CRISPR TYPE V SYSTEMS CARIBOU BIOSCIENCES, INC. (US) 2023-10-19 WO claimed
EP-3668867-B1 SYNTHESIS, PHARMACOLOGY AND USE OF NEW AND SELECTIVE FMS-LIKE TYROSINE KINASE 3 (FLT3) FLT3 INHIBITORS UNIV REGENSBURG (DE) 2023-10-04 EP claimed
EP-3071040-B2 METHOD FOR SCALABLE SKELETAL MUSCLE LINEAGE SPECIFICATION AND CULTIVATION UNIV MISSOURI (US) 2022-12-28 EP claimed
US-20210177760-A1 DRUG DELIVERY COMPOSITION AND METHOD OF FABRICATION DIGNITY HEALTH 2021-06-17 US claimed
EP-2797898-B9 PIPERAZINYL DERIVATIVES FOR THE TREATMENT OF CANCERS PITTY MARC HENRY (FR) 2021-05-26 EP claimed
WO-2021069690-A1 FILM THAI POLYETHYLENE CO., LTD. (TH) 2021-04-15 WO claimed
EP-3283463-B1 DIMERIC QUINACRINE DERIVATIVES AS AUTOPHAGY INHIBITORS FOR CANCER THERAPY UNIV PENNSYLVANIA (US) 2021-01-20 EP claimed
WO-2020231937-A1 IRF2 AS A PROGNOSTIC BIOMARKER AND TARGET FOR AUGMENTING IMMUNOTHERAPY UNIVERSITY OF MASSACHUSETTS (US) 2020-11-19 WO claimed
EP-3328185-B1 METHOD FOR PRODUCING HAPLOID, DIHAPLOID AND DOUBLED HAPLOID PLANTS BY ISOLATED MICROSPORE CULTURE VILMORIN & CIE (FR) 2020-06-24 EP claimed
JP-2007504131-A 2007-03-01 JP claimed
EP-1667680-A2 COMBINATION METHODS OF TREATING CANCER Aton Pharma, Inc. (US) 2006-06-14 EP claimed
EP-1545536-A2 METHOD OF TREATING LEUKEMIA WITH A COMBINATION OF SUBEROYLANILIDE HYDROMAXIC ACID AND IMATINIB MESYLATE UNIVERSITY OF SOUTH FLORIDA (US) 2005-06-29 EP claimed
WO-2005023179-A2 COMBINATION METHODS OF TREATING CANCER ATON PHARMA, INC. (US) 2005-03-17 WO claimed
EP-1297851-B1 Inhibition of histone deacetylase as a treatment for cardiac hypertrophy UNIV COLORADO (US) 2005-01-26 EP claimed
US-20040127571-A1 Method of Treating Leukemia with a Combination of Suberoylanilide Hydromaxic Acid and Imatinib Mesylate UNIVERSITY OF SOUTH FLORIDA (US) 2004-07-01 US claimed
WO-2004026234-A2 METHOD OF TREATING LEUKEMIA WITH A COMBINATION OF SUBEROYLANILIDE HYDROMAXIC ACID AND IMATINIB MESYLATE UNIVERSITY OF SOUTH FLORIDA (US) 2004-04-01 WO claimed
WO-2002055017-A2 METHOD OF TREATING AUTOIMMUNE DISEASES WAKE FOREST UNIVERSITY (US) 2002-07-18 WO claimed
US-6235823-B1 CRYSTALLINE POLYPROPLYLENE RESIN AND A BETA-NUCLEATING AGENT, THE BETA-NUCLEATING AGENT BEING A DIAMIDE COMPOUND. NEW JAPAN CHEMICAL CO., LTD. (JP) 2001-05-22 US claimed
EP-0557721-A2 Crystalline polypropylene resin composition and amide compounds NEW JAPAN CHEMICAL CO.,LTD. (JP) 1993-09-01 EP claimed