SCHEMBL13735129

SCHEMBL13735129

Cn1cc(Nc2ncc3cc[nH]c3n2)cn1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 10/20 0.53
JAK2 O60674 9/20 0.53
JAK3 P52333 6/20 0.53
TYK2 P29597 6/20 0.53
ALK Q9UM73 5/20 0.51
CDK19 Q9BWU1 4/20 0.51
LRRK2 Q5S007 1/20 0.49
PTK2 Q05397 1/20 0.48
MAPK1 P28482 1/20 0.47
EGFR P00533 1/20 0.44
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
INCENP Q9NQS7 1/20 0.44
TPX2 Q9ULW0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29979953 0.80 JAK1 (0.50) JAK1JAK2JAK3TYK2ALK
SCHEMBL672922 0.79 JAK1 (0.52) JAK1JAK2JAK3TYK2ALK
SCHEMBL22159389 0.78 APP (0.50) JAK1JAK2JAK3TYK2ALK
SCHEMBL14801269 0.77 PTK2 (0.56) JAK1JAK2JAK3ALKCDK19
SCHEMBL14801718 0.77 PTK2 (0.56) JAK1JAK2JAK3ALKCDK19
SCHEMBL19027053 0.76 PTK2 (0.64) JAK3ALKCDK19LRRK2PTK2
SCHEMBL15380926 0.75 CDK2 (0.54) JAK2JAK3TYK2LRRK2PTK2
SCHEMBL29813554 0.75 EGFR (0.62) ALKEGFRAURKA
SCHEMBL17112501 0.74 EGFR (0.48) PTK2EGFR
SCHEMBL6882453 0.73 AURKA (0.55) MAPK1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012143320-A1 (7H-PYRROLO[2,3-D]PYRIMIDIN-2-YL)AMINE COMPOUNDS AS JAK3 INHIBITORS CELLZOME LIMITED (GB) 2012-10-26 WO disclosed