SCHEMBL13740912

SCHEMBL13740912

Nc1ccc2c(c1I)CCN(C(=O)O)C2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.35
NOTUM Q6P988 1/20 0.34
AKR1C3 P42330 2/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
ABHD6 Q9BV23 4/20 0.33
HDAC8 Q9BY41 1/20 0.32
ESR1 P03372 4/20 0.32
ESR2 Q92731 4/20 0.32
TMPRSS2 O15393 2/20 0.32
BTK Q06187 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16961694 0.82 ABHD6 (0.37) NR1H2NOTUMAKR1C3NPC1TP53
SCHEMBL28534853 0.82 ABHD6 (0.35) NR1H2NOTUMAKR1C3NPC1TP53
SCHEMBL13739622 0.80 NR1H2 (0.60) NR1H2MAPTESR2KDM4E
SCHEMBL16962869 0.78 BPTF (0.41) NR1H2SMN1; SMN2MEN1MAPTKMT2A
SCHEMBL16111044 0.78 AKR1C3 (0.51) NOTUMAKR1C3NPC1TP53RAB9A
SCHEMBL17607348 0.73 RAC1 (0.38) NOTUMNPC1TP53RAB9ASMN1; SMN2
SCHEMBL29150707 0.73 ABHD6 (0.37) NR1H2NOTUMNPC1TP53RAB9A
SCHEMBL29372803 0.72 NOTUM (0.33) NOTUMNPC1TP53RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL8384089 0.72 KDM4E (0.45) NOTUMNPC1TP53RAB9ASMN1; SMN2
SCHEMBL31447535 0.71 ITGB2 (0.35) NR1H2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022022489-A1 INDOLE FUSED RING DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE 江苏恒瑞医药股份有限公司 2022-02-03 WO disclosed
WO-2012154888-A1 COMPOUNDS FOR TREATING PROTEIN FOLDING DISORDERS PROTEOSTASIS THERAPEUTICS, INC. (US) 2012-11-15 WO disclosed