SCHEMBL28534853

SCHEMBL28534853

Nc1ccc2c(c1F)CCN(C(=O)O)C2

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 5/20 0.35
ESR1 P03372 5/20 0.35
ESR2 Q92731 5/20 0.35
NR1H2 P55055 1/20 0.35
NOTUM Q6P988 1/20 0.34
NPC1 O15118 4/20 0.33
RAB9A P51151 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
AKR1C3 P42330 1/20 0.33
TP53 P04637 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HDAC8 Q9BY41 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13740912 0.82 NR1H2 (0.35) ABHD6ESR1ESR2NR1H2NOTUM
SCHEMBL16961694 0.82 ABHD6 (0.37) ABHD6ESR1ESR2NR1H2NOTUM
SCHEMBL20162141 0.82 ABHD6 (0.42) ABHD6ESR1ESR2NOTUMNPC1
SCHEMBL31067476 0.80 NR1H2 (0.60) ABHD6ESR2NR1H2MAPTALDH1A1
SCHEMBL4165540 0.80 NR1H2 (0.60) ABHD6ESR2NR1H2MAPTALDH1A1
SCHEMBL22981183 0.79 KCNJ1 (0.37) ABHD6ESR1ESR2NOTUMNPC1
SCHEMBL30597676 0.79 ABHD6 (0.36) ABHD6ESR1ESR2NOTUMNPC1
SCHEMBL16962869 0.78 BPTF (0.41) ABHD6NR1H2SMN1; SMN2MEN1MAPT
SCHEMBL16111044 0.78 AKR1C3 (0.51) ABHD6NOTUMNPC1RAB9ASMN1; SMN2
SCHEMBL27771947 0.77 HTR5A (0.42) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307772-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2024-06-28 CN disclosed
CN-113307772-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-08-27 CN disclosed
CN-106257976-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-02-02 CN disclosed