SCHEMBL13740985

SCHEMBL13740985

CCOC(=O)c1c(O)c2c(=O)n(C)c3ccccc3c2n1C

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.64
KDM4E B2RXH2 5/20 0.64
NPC1 O15118 1/20 0.54
ALOX15 P16050 1/20 0.54
HSD17B10 Q99714 2/20 0.52
TSHR P16473 1/20 0.52
RXFP1 Q9HBX9 2/20 0.50
LMNA P02545 2/20 0.49
RECQL P46063 1/20 0.48
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
PABPC1 P11940 1/20 0.46
KMT2A Q03164 1/20 0.46
HPGD P15428 1/20 0.46
GABRP O00591 1/20 0.45
GABRD O14764 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13739731 0.86 ALDH1A1 (0.55) ALDH1A1KDM4ENPC1ALOX15HSD17B10
SCHEMBL1062395 0.85 KDM4E (0.51) ALDH1A1KDM4ENPC1ALOX15HSD17B10
SCHEMBL9867870 0.82 ALDH1A1 (0.68) ALDH1A1KDM4ENPC1ALOX15HSD17B10
SCHEMBL1062493 0.81 FEN1 (0.51) ALDH1A1KDM4ERXFP1LMNARECQL
SCHEMBL30099678 0.78 ALDH1A1 (1.00) ALDH1A1KDM4ENPC1ALOX15HSD17B10
SCHEMBL14829909 0.78 ALDH1A1 (0.80) ALDH1A1KDM4ENPC1ALOX15HSD17B10
SCHEMBL1061607 0.78 ALDH1A1 (1.00) ALDH1A1KDM4ENPC1ALOX15HSD17B10
SCHEMBL13708824 0.77 ALDH1A1 (0.42) ALDH1A1KDM4ENPC1ALOX15HSD17B10
SCHEMBL1060211 0.76 HSD17B10 (0.61) ALDH1A1KDM4ENPC1ALOX15HSD17B10
SCHEMBL30639225 0.74 TSHR (0.66) ALDH1A1KDM4ENPC1ALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012154731-A1 SUBSTITUTED 1H-PYRROLO[3,2-C]QUINOLIN-4(5H)-ONE ANALOGS AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2012-11-15 WO disclosed
WO-2012154731-A1 SUBSTITUTED 1H-PYRROLO[3,2-C]QUINOLIN-4(5H)-ONE ANALOGS AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2012-11-15 WO disclosed