SCHEMBL13739731

SCHEMBL13739731

CCOC(=O)c1c(OC)c2c(=O)n(C)c3ccccc3c2n1C

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 3/20 0.55
RXFP1 Q9HBX9 2/20 0.51
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50
NPC1 O15118 1/20 0.47
ALOX15 P16050 1/20 0.47
MAPK1 P28482 1/20 0.46
MAPT P10636 1/20 0.45
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
PABPC1 P11940 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13740985 0.86 ALDH1A1 (0.64) ALDH1A1KDM4ERXFP1TSHRHSD17B10
SCHEMBL1055219 0.85 KMT2A (0.48) ALDH1A1KDM4ERXFP1MAPK1MEN1
SCHEMBL13740053 0.85 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10PABPC1KMT2A
SCHEMBL1061698 0.84 KMT2A (0.50) ALDH1A1KDM4ERXFP1MAPTMEN1
SCHEMBL9868002 0.82 ALDH1A1 (0.54) ALDH1A1KDM4ERXFP1TSHRHSD17B10
SCHEMBL752911 0.82 ALDH1A1 (0.57) ALDH1A1KDM4ERXFP1TSHRHSD17B10
SCHEMBL1057049 0.78 KMT2A (0.48) ALDH1A1KDM4ERXFP1MAPTMEN1
SCHEMBL1059735 0.77 TSHR (0.59) ALDH1A1KDM4ERXFP1TSHRHSD17B10
SCHEMBL13838736 0.76 RXFP1 (0.52) ALDH1A1KDM4ERXFP1TSHRHSD17B10
SCHEMBL1063196 0.75 KMT2A (0.45) ALDH1A1RXFP1MAPTMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012154731-A1 SUBSTITUTED 1H-PYRROLO[3,2-C]QUINOLIN-4(5H)-ONE ANALOGS AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2012-11-15 WO disclosed