SCHEMBL13745159

SCHEMBL13745159

CCc1ccc(-c2ccc(C)cn2)cn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.52
CCR5 P51681 1/20 0.52
CCR8 P51685 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
CYP3A4 P08684 1/20 0.50
CYP2A6 P11509 1/20 0.50
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
METAP2 P50579 1/20 0.40
PTGS2 P35354 3/20 0.38
PTGS1 P23219 1/20 0.38
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
PDE10A Q9Y233 1/20 0.38
GRIA2 P42262 1/20 0.37
KDM1A O60341 1/20 0.37
LMNA P02545 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL469189 0.84
SCHEMBL14804380 0.82 CCR1 (0.76) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL13745161 0.81 NPC1 (0.42) NPC1RAB9ASMN1; SMN2PTGS2PTGS1
SCHEMBL17051522 0.81 CCR1 (0.65) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL17051514 0.78 CCR1 (0.75) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL26040044 0.78 PRMT5 (0.46) PTGS2PTGS1PRMT5WDR77PDE10A
SCHEMBL8233550 0.78 CCR1 (0.56) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL3426229 0.77 CYP3A4 (0.61) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL17051547 0.77 CCR1 (0.60) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL2477927 0.76 CCR1 (0.71) CCR1CCR5CCR8HDAC6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095377-A1 SPIRO COMPOUNDS AS NPY Y5 RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-08-06 WO disclosed