SCHEMBL13745161

SCHEMBL13745161

CCc1ccc(-c2ccc(F)cn2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RXFP1 Q9HBX9 1/20 0.42
BRS3 P32247 3/20 0.40
GRM5 P41594 3/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GRIA2 P42262 3/20 0.39
KCNH2 Q12809 2/20 0.39
AURKA O14965 1/20 0.38
ABL1 P00519 1/20 0.38
NTRK1 P04629 1/20 0.38
LCK P06239 1/20 0.38
CSF1R P07333 1/20 0.38
RET P07949 1/20 0.38
MET P08581 1/20 0.38
PDGFRB P09619 1/20 0.38
PIM1 P11309 1/20 0.38
PDGFRA P16234 1/20 0.38
FLT3 P36888 1/20 0.38
MAPK8 P45983 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2336915 0.85
SCHEMBL22186144 0.82 PRMT5 (0.40) NPC1GRM5RAB9ASMN1; SMN2KCNH2
SCHEMBL13745159 0.81 CCR1 (0.52) NPC1RAB9ASMN1; SMN2GRIA2AURKA
SCHEMBL3823523 0.80 GRM5 (0.41) NPC1RXFP1BRS3GRM5GRIA2
SCHEMBL3823318 0.79 RAB9A (0.53) NPC1RXFP1BRS3RAB9ASMN1; SMN2
SCHEMBL26040044 0.77 PRMT5 (0.46) PTGS1PTGS2PRMT5WDR77
SCHEMBL13750539 0.77 TDO2 (0.46) NPC1RXFP1BRS3GRM5GRIA2
SCHEMBL7945448 0.74 MMP13 (0.42)
SCHEMBL12533576 0.74 CYP1A2 (0.50) NPC1BRS3GRM5RAB9ASMN1; SMN2
SCHEMBL4024197 0.73 TDO2 (0.46) NPC1RXFP1RAB9APTPN1PTPN6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095377-A1 SPIRO COMPOUNDS AS NPY Y5 RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-08-06 WO disclosed