SCHEMBL13745641

SCHEMBL13745641

CCc1cccc(-c2cc(F)ccc2N)n1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.39
TGFBR1 P36897 6/20 0.38
CCNE1 P24864 2/20 0.35
CDK2 P24941 2/20 0.35
CCNE2 O96020 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GRM5 P41594 3/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
TLR8 Q9NR97 1/20 0.33
NPC1 O15118 1/20 0.33
CHRNA7 P36544 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10304946 0.83 CTSA (0.43) KCNH2TGFBR1GRM5
SCHEMBL22841384 0.81 TRPV3 (0.43) TGFBR1ALDH1A1TLR8
SCHEMBL13745259 0.76 NPC1 (0.42) TGFBR1CCNE1CDK2CCNE2ALDH1A1
SCHEMBL13745269 0.76 HSP90AA1 (0.50) HSP90AA1HSP90AB1
SCHEMBL20878875 0.74 MAP4K4 (0.47) TLR8KDM4EMEN1MAPTKMT2A
SCHEMBL996802 0.74 NOS2 (0.41) TGFBR1CCNE1CDK2ALDH1A1GRM5
SCHEMBL13534470 0.74 SCN9A (0.46) TGFBR1ALDH1A1TLR8NPC1MEN1
SCHEMBL6205528 0.73 SMN1; SMN2 (0.39) CCNE1CDK2CCNE2ALDH1A1NPC1
SCHEMBL244011 0.72 CCR1 (0.46) KCNH2TGFBR1CCNE1CDK2HSP90AA1
SCHEMBL19091155 0.71 CYP1A2 (0.35) KCNH2TGFBR1KDM4EMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009097578-A1 OXIM DERIVATIVES AS HSP90 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-08-06 WO disclosed