SCHEMBL13748418

SCHEMBL13748418

O=C(O)c1cc(Cl)c(Cl)cc1C(=O)N1CCc2c([nH]c3ccccc23)C1c1ccc(F)c(-c2nnn[nH]2)c1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 15/20 0.57
ABCB1 P08183 9/20 0.57
LMNA P02545 2/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
NPSR1 Q6W5P4 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13749166 0.79 KDM4E (0.47) ABCG2ABCB1LMNAMAPTNPSR1
SCHEMBL13748440 0.76 MAPT (0.66) ABCG2MAPTNPSR1MAPK1
SCHEMBL13882262 0.73 ABCG2 (0.71) ABCG2ABCB1LMNAMAPTNPSR1
SCHEMBL13882337 0.73 ABCG2 (0.74) ABCG2ABCB1LMNATP53MAPT
SCHEMBL13749167 0.72 MAPT (0.47) ABCG2ABCB1LMNAMAPTNPSR1
SCHEMBL13748742 0.72 TSHR (0.59) ABCG2ABCB1LMNA
SCHEMBL13882446 0.72 ABCG2 (0.89) ABCG2ABCB1LMNATP53NPSR1
SCHEMBL13882509 0.72 ABCG2 (0.81) ABCG2ABCB1LMNATP53
SCHEMBL4264083 0.70 ABCG2 (1.00) ABCG2ABCB1LMNANPSR1SMN1; SMN2
SCHEMBL13882344 0.70 LMNA (0.70) ABCG2ABCB1LMNATP53NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009102377-A2 ANTIBIOTIC TETRAHYDRO-BETA-CARBOLINE DERIVATIVES MAXTHERA INC. (US) 2009-08-20 WO disclosed