SCHEMBL13748883

SCHEMBL13748883

C=CNc1ccc2[nH]nc(-c3ccc(OC(C)C)nc3)c2c1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.61
MAPK1 P28482 4/20 0.46
MET P08581 1/20 0.45
NTRK1 P04629 1/20 0.43
KDR P35968 1/20 0.41
ETV6 P41212 1/20 0.41
MAPK3 P27361 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11996741 0.89 LRRK2 (0.61) LRRK2MAPK1METNTRK1KDR
SCHEMBL20420387 0.79 LRRK2 (0.52) LRRK2MAPK1METKDRETV6
SCHEMBL13495128 0.79 LRRK2 (0.52) LRRK2MAPK1METKDRETV6
SCHEMBL27852657 0.76 MAPK1 (0.53) LRRK2MAPK1MET
SCHEMBL29643985 0.76 LRRK2 (1.00) LRRK2
SCHEMBL22890316 0.76 LRRK2 (1.00) LRRK2
SCHEMBL23207731 0.72 NTRK1 (0.52) LRRK2MAPK1NTRK1MAPK3
SCHEMBL2277926 0.72 LRRK2 (0.57) LRRK2MAPK1MAPK3
SCHEMBL11996761 0.72 LRRK2 (0.57) LRRK2MAPK1MAPK3
SCHEMBL17144260 0.72 LRRK2 (0.57) LRRK2MAPK1METMAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009105500-A1 COMPOUNDS THAT ARE ERK INHIBITORS SCHERING CORPORATION (US) 2009-08-27 WO disclosed