SCHEMBL13748972

SCHEMBL13748972

CCOc1cc(-c2nn(C(c3ccccc3)(c3ccccc3)c3ccccc3)c3ccc(NCO)cc23)ccn1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACSS2 Q9NR19 2/20 0.33
PTGER2 P43116 1/20 0.33
KIT P10721 1/20 0.32
PTGER1 P34995 1/20 0.31
NTRK1 P04629 1/20 0.31
CDK2 P24941 1/20 0.31
GSK3B P49841 1/20 0.31
MAPK1 P28482 1/20 0.30
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748615 0.92 LRRK2 (0.37) ACSS2MAPK1LRRK2
SCHEMBL13749233 0.89 MAPK1 (0.33) KITMAPK1
SCHEMBL2274094 0.84 CNR1 (0.36) ACSS2KITPTGER1NTRK1MAPK1
SCHEMBL2276520 0.80 L3MBTL1 (0.47)
SCHEMBL17146107 0.75 MAPK1 (0.33) KITMAPK1LRRK2
SCHEMBL12374202 0.74 MAPK1 (0.41) MAPK1
SCHEMBL2277546 0.74 MAPK1 (0.41) MAPK1
SCHEMBL17430340 0.74 TTK (0.41) ACSS2PTGER1NTRK1
SCHEMBL2280858 0.73 CNR1 (0.35) KITPTGER1MAPK1LRRK2
SCHEMBL30084146 0.71 PTGER1 (0.41) PTGER1NTRK1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009105500-A1 COMPOUNDS THAT ARE ERK INHIBITORS SCHERING CORPORATION (US) 2009-08-27 WO disclosed