SCHEMBL13748615

SCHEMBL13748615

COc1cc(-c2nn(C(c3ccccc3)(c3ccccc3)c3ccccc3)c3ccc(NCO)cc23)ccn1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.37
WNT3A P56704 1/20 0.35
MAPK1 P28482 2/20 0.34
CNR1 P21554 1/20 0.34
ATR Q13535 1/20 0.33
MET P08581 2/20 0.32
BUB1 O43683 1/20 0.32
MAPT P10636 1/20 0.32
DGAT2 Q96PD7 1/20 0.32
DYRK1A Q13627 1/20 0.32
ACSS2 Q9NR19 1/20 0.32
ROCK2 O75116 1/20 0.31
SLC13A5 Q86YT5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748972 0.92 ACSS2 (0.33) LRRK2MAPK1ACSS2
SCHEMBL13749233 0.90 MAPK1 (0.33) MAPK1
SCHEMBL2280858 0.82 CNR1 (0.35) LRRK2MAPK1CNR1ATRDYRK1A
SCHEMBL2276443 0.78 L3MBTL1 (0.49) CNR1MAPT
SCHEMBL31021936 0.77 MAPK1 (0.34) LRRK2MAPK1BUB1DYRK1AROCK2
SCHEMBL17146107 0.75 MAPK1 (0.33) LRRK2MAPK1MAPT
SCHEMBL2274094 0.75 CNR1 (0.36) MAPK1CNR1MAPTACSS2
SCHEMBL12374195 0.73 JAK2 (0.37) MAPK1METBUB1DGAT2
SCHEMBL2273869 0.73 JAK2 (0.37) MAPK1METBUB1DGAT2
SCHEMBL30084146 0.72 PTGER1 (0.41) LRRK2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009105500-A1 COMPOUNDS THAT ARE ERK INHIBITORS SCHERING CORPORATION (US) 2009-08-27 WO disclosed