SCHEMBL1375388

SCHEMBL1375388

Nc1ncc(Oc2ccc(Cl)cc2)c(NCC2CCC(O)C2)n1.Nc1ncc(Oc2ccc(Cl)cc2)c(NCC2CCCC2O)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 3/20 0.36
CNR2 P34972 2/20 0.33
EGLN1 Q9GZT9 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
TNK2 Q07912 1/20 0.32
IRAK1 P51617 5/20 0.32
IDO1 P14902 2/20 0.32
TRPC6 Q9Y210 1/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
PRKCQ Q04759 1/20 0.30
CCNT1 O60563 1/20 0.30
CCNC P24863 1/20 0.30
CDK8 P49336 1/20 0.30
CDK9 P50750 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30
CNR1 P21554 1/20 0.30
KCNH2 Q12809 2/20 0.30
SCN9A Q15858 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1375389 1.00 TDO2 (0.36) TDO2CNR2EGLN1NOS3NOS1
SCHEMBL1375711 0.96 TDO2 (0.37) TDO2CNR2EGLN1NOS3NOS1
SCHEMBL1375708 0.96 TDO2 (0.37) TDO2CNR2EGLN1NOS3NOS1
SCHEMBL5203028 0.92 IRAK1 (0.36) EGLN1NOS3NOS1IRAK1TRPC6
SCHEMBL1376037 0.92 IRAK1 (0.36) EGLN1NOS3NOS1IRAK1TRPC6
SCHEMBL1376032 0.92 IRAK1 (0.36) EGLN1NOS3NOS1IRAK1TRPC6
SCHEMBL5206015 0.92 TDO2 (0.41) TDO2CNR2EGLN1NOS3NOS1
SCHEMBL1376197 0.92 TDO2 (0.41) TDO2CNR2EGLN1NOS3NOS1
SCHEMBL1376035 0.92 IRAK1 (0.36) EGLN1NOS3NOS1IRAK1TRPC6
SCHEMBL5203021 0.92 IRAK1 (0.36) EGLN1NOS3NOS1IRAK1TRPC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4743463-B2 2011-08-10 JP claimed
JP-2002541245-A 2002-12-03 JP claimed
EP-1165523-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP claimed
WO-2000061562-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-19 WO claimed
EP-1165523-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000061562-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-19 WO disclosed