SCHEMBL1375708

SCHEMBL1375708

Nc1ncc(Oc2ccc(Cl)cc2)c(NCC2CCCC(O)C2)n1.Nc1ncc(Oc2ccc(Cl)cc2)c(NCC2CCCCC2O)n1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 3/20 0.37
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
IRAK1 P51617 3/20 0.34
IDO1 P14902 2/20 0.33
CNR2 P34972 1/20 0.33
APP P05067 1/20 0.32
TNK2 Q07912 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
TLR7 Q9NYK1 1/20 0.30
CHEK1 O14757 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1375711 1.00 TDO2 (0.37) TDO2NOS3NOS1EGLN1IRAK1
SCHEMBL1375389 0.96 TDO2 (0.36) TDO2NOS3NOS1EGLN1IRAK1
SCHEMBL1375388 0.96 TDO2 (0.36) TDO2NOS3NOS1EGLN1IRAK1
SCHEMBL1378803 0.93 IRAK1 (0.38) NOS3NOS1EGLN1IRAK1APP
SCHEMBL1378801 0.93 IRAK1 (0.38) NOS3NOS1EGLN1IRAK1APP
SCHEMBL5205868 0.93 IRAK1 (0.38) NOS3NOS1EGLN1IRAK1APP
SCHEMBL5205876 0.93 IRAK1 (0.38) NOS3NOS1EGLN1IRAK1APP
SCHEMBL1378800 0.93 IRAK1 (0.38) NOS3NOS1EGLN1IRAK1APP
SCHEMBL1377884 0.91 TDO2 (0.43) TDO2NOS3NOS1EGLN1IRAK1
SCHEMBL5206015 0.91 TDO2 (0.41) TDO2NOS3NOS1EGLN1IRAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4743463-B2 2011-08-10 JP claimed
JP-2002541245-A 2002-12-03 JP claimed
EP-1165523-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP claimed
WO-2000061562-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-19 WO claimed
EP-1165523-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000061562-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-19 WO disclosed