SCHEMBL13763556

SCHEMBL13763556

N#Cc1c[nH]c2ccc(CCCN3CCN(c4ccc5c(c4)CC(C(N)=O)O5)CC3)cc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.46
ADRA2A P08913 3/20 0.46
ADRA2C P18825 3/20 0.46
ADRA1D P25100 3/20 0.46
ADRA1A P35348 3/20 0.46
ADRA1B P35368 3/20 0.46
SLC6A2 P23975 3/20 0.46
SLC6A4 P31645 3/20 0.46
SLC6A3 Q01959 3/20 0.46
DRD2 P14416 2/20 0.46
HTR7 P34969 2/20 0.46
ADRA2B P18089 2/20 0.46
KCNH2 Q12809 1/20 0.46
ADRB2 P07550 1/20 0.46
DRD4 P21917 1/20 0.46
FPR3 P25089 1/20 0.46
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46
GPR183 P32249 1/20 0.46
HRH1 P35367 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16578994 0.82 HTR1A (0.68) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL1323756 0.80 HTR1A (0.70) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL1323812 0.80 HTR1A (0.65) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL1322969 0.78 HTR1A (0.57) HTR1AHTR1DHTR1B
SCHEMBL1406042 0.77 HTR1A (0.57) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL13633559 0.77 ADRA2A (0.48) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL27480588 0.76 HTR1A (0.68) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL1323781 0.75 HTR1A (0.43) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL1323787 0.75 HTR1A (0.53) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL1322976 0.75 HTR1A (0.51) HTR1AADRA2AADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7572796-B2 Substituted indoles MERCK PATENT GMBH (DE) 2009-08-11 US disclosed