SCHEMBL13765504

SCHEMBL13765504

COCc1c(-c2nc(-c3ccc(CN4C=NCN4)cc3)no2)nnn1-c1ccccc1F

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 7/20 0.38
MAPT P10636 7/20 0.38
RXFP1 Q9HBX9 1/20 0.36
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
GLA P06280 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 2/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
S1PR1 P21453 5/20 0.34
LMNA P02545 1/20 0.34
S1PR3 Q99500 3/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10182852 0.86 TP53 (0.42) TP53MAPTRXFP1ALDH1A1SMN1; SMN2
SCHEMBL10181578 0.84 MAPT (0.53) TP53MAPTRXFP1ALDH1A1SMN1; SMN2
SCHEMBL3455783 0.83 TP53 (0.43) TP53MAPTRXFP1ALDH1A1SMN1; SMN2
SCHEMBL3756827 0.83 TP53 (0.41) TP53MAPTRXFP1ALDH1A1SMN1; SMN2
SCHEMBL3763187 0.83 MAPT (0.49) TP53MAPTRXFP1ALDH1A1SMN1; SMN2
SCHEMBL3758471 0.82 S1PR1 (0.39) TP53MAPTRXFP1SMN1; SMN2NPC1
SCHEMBL10179530 0.81 TP53 (0.54) TP53MAPTALDH1A1SMN1; SMN2HSD17B10
SCHEMBL3766224 0.81 MAOA (0.43) TP53MAPTRXFP1ALDH1A1SMN1; SMN2
SCHEMBL10179953 0.80 RAB9A (0.47) TP53MAPTSMN1; SMN2HSD17B10NPC1
SCHEMBL27829115 0.79 TP53 (0.45) TP53MAPTRXFP1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080663-A1 TRIAZOLE OXADIAZOLES DERIVATIVES MERCK SERONO S.A. (CH) 2009-07-02 WO disclosed