SCHEMBL13765865

SCHEMBL13765865

C#Cc1cncc2c(C)cccc12

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.44
CYP2A6 P11509 3/20 0.44
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
RAF1 P04049 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
PSMD14 O00487 1/20 0.31
COPS5 Q92905 1/20 0.31
MAPT P10636 1/20 0.31
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404557 0.77 CYP1A2 (0.62) CYP1A2CYP2A6ALDH1A1HPGDHSD17B10
SCHEMBL4064172 0.77 ALDH1A1 (0.44) CYP1A2ALDH1A1HPGDHSD17B10NCOA3
SCHEMBL13765864 0.72 CYP1A2 (0.48) CYP1A2CYP2A6ALDH1A1HPGDHSD17B10
SCHEMBL19663002 0.72 CYP1A2 (0.48) CYP1A2CYP2A6ALDH1A1HPGDHSD17B10
SCHEMBL19953988 0.72 CYP1A2 (0.48) CYP1A2CYP2A6ALDH1A1HPGDHSD17B10
SCHEMBL2203417 0.71 CYP1A2 (0.59) CYP1A2CYP2A6ALDH1A1HPGDHSD17B10
SCHEMBL4062748 0.69 HTT (0.44) CYP1A2CYP11B1CYP11B2
SCHEMBL19660435 0.69 CYP2A6 (0.44) CYP1A2CYP2A6ALDH1A1HPGD
SCHEMBL19660419 0.69 CYP1A2 (0.44) CYP1A2CYP2A6ALDH1A1MAPTCYP11B1
SCHEMBL19660438 0.69 CYP2A6 (0.44) CYP1A2CYP2A6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8461167-B2 Acetylenic heteroaryl compounds ARIAD PHARMACEUTICALS, INC. (US) 2013-06-11 US disclosed
US-20090176781-A1 Acetylenic Heteroaryl Compounds ARIAD PHARMACEUTICALS, INC. 2009-07-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176781-A1 Acetylenic Heteroaryl Compounds NAT1, AADAC, ACACA CYP1A2 32/4885CYP2A6 61/4885ALDH1A1 148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.