SCHEMBL1377129

SCHEMBL1377129

CCC(C(=O)OCC(C)C)N(CC1CC1)c1ccc(C#N)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PGR P06401 20/20 0.47
CYP2C19 P33261 4/20 0.47
CYP2C9 P11712 8/20 0.39
CYP2D6 P10635 7/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1379962 0.91 PGR (0.37) PGRCYP2C19
SCHEMBL1376889 0.86 PGR (0.48) PGRCYP2C19CYP2C9CYP2D6KCNH2
SCHEMBL1376545 0.86 PGR (0.48) PGRCYP2C19CYP2C9CYP2D6KCNH2
SCHEMBL1377127 0.86 PGR (0.45) PGRCYP2C19CYP2C9CYP2D6KCNH2
SCHEMBL1377211 0.84 PGR (0.46) PGRCYP2C19CYP2C9CYP2D6KCNH2
SCHEMBL1379593 0.83 PGR (0.46) PGRCYP2C19CYP2C9CYP2D6KCNH2
SCHEMBL1380583 0.83 PGR (0.48) PGRCYP2C19CYP2C9CYP2D6
SCHEMBL1377099 0.81 PGR (0.42) PGRCYP2C19CYP2C9CYP2D6KCNH2
SCHEMBL1377609 0.80 PGR (0.52) PGRCYP2C19CYP2C9CYP2D6KCNH2
SCHEMBL1377611 0.80 PGR (0.52) PGRCYP2C19CYP2C9CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4805909-B2 2011-11-02 JP claimed
EP-1725522-A1 ANILINE DERIVATIVES AS SELECTIVE ANDROGEN RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-29 EP claimed
WO-2005085185-A1 ANILINE DERIVATIVES AS SELECTIVE ANDROGEN RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-15 WO claimed
EP-1725522-A1 ANILINE DERIVATIVES AS SELECTIVE ANDROGEN RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-29 EP disclosed
WO-2005085185-A1 ANILINE DERIVATIVES AS SELECTIVE ANDROGEN RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-15 WO disclosed