SCHEMBL13777

SCHEMBL13777

O=CC[C@@H]1C[C@H]1c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 11/20 0.57
MAOB P27338 9/20 0.57
HTR2B P41595 6/20 0.57
HTR2A P28223 4/20 0.57
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
MAOA P21397 7/20 0.43
KDM1A O60341 5/20 0.43
CYP2C19 P33261 4/20 0.43
CYP2B6 P20813 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
TAAR1 Q96RJ0 2/20 0.43
LMNA P02545 1/20 0.43
CYP3A4 P08684 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2A6 P11509 1/20 0.43
SLC6A2 P23975 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25254330 1.00 HTR2C (0.57) HTR2CMAOBHTR2BHTR2ADRD2
SCHEMBL13778 1.00 HTR2C (0.57) HTR2CMAOBHTR2BHTR2ADRD2
SCHEMBL6560505 0.81 HTR2C (0.53) HTR2CMAOBHTR2BHTR2ADRD2
SCHEMBL6250926 0.81 KDM1A (0.43) HTR2CMAOBHTR2BHTR2ADRD2
SCHEMBL3395704 0.80 HTR2C (0.57) HTR2CMAOBHTR2BHTR2ADRD2
SCHEMBL6584873 0.80 HTR2C (0.57) HTR2CMAOBHTR2BHTR2ADRD2
SCHEMBL10675977 0.79 MEN1 (0.42) HTR2CMAOBHTR2BHTR2AMAOA
SCHEMBL10675972 0.79 MEN1 (0.42) HTR2CMAOBHTR2BHTR2AMAOA
SCHEMBL6406073 0.79 MEN1 (0.42) HTR2CMAOBHTR2BHTR2AMAOA
SCHEMBL10676736 0.79 MEN1 (0.42) HTR2CMAOBHTR2BHTR2AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed