SCHEMBL13788560

SCHEMBL13788560

O=C(O)c1n[nH]c2c1COc1cc(N3CC[C@H](O)C3)ccc1-2

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.38
ABL1 P00519 1/20 0.37
SLC40A1 Q9NP59 1/20 0.36
CHEK1 O14757 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ALPL P05186 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CDK1 P06493 1/20 0.35
CDK2 P24941 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
PRKAG1 P54619 2/20 0.35
PRKAA1 Q13131 2/20 0.35
PRKAB1 Q9Y478 2/20 0.35
HCAR2 Q8TDS4 1/20 0.34
PRKAB2 O43741 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3521482 0.86 IDH1 (0.40) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
Hydrochloric Acid SCHEMBL3519180 0.85 IDH1 (0.39) PRKAG1PRKAA1PRKAB1PRKAB2PRKAA2
SCHEMBL3520429 0.76 HCAR2 (0.41) ARKDM4EALDH1A1ALPLHSD17B10
SCHEMBL2171482 0.75 KDM4E (0.59) KDM4EALDH1A1ALPLHSD17B10HCAR2
SCHEMBL3747711 0.73 KMT2A (0.44) KDM4EALDH1A1ALPLHSD17B10PRKAG1
SCHEMBL13788543 0.73 UGCG (0.42) ALPLCDK2
SCHEMBL3518362 0.73 UGCG (0.41)
SCHEMBL3518121 0.68 ALDH1A1 (0.43) ARKDM4EALDH1A1ALPLHSD17B10
SCHEMBL4728060 0.68 ALPL (0.43) KDM4EALDH1A1ALPLHSD17B10PRKAG1
SCHEMBL3518546 0.68 MAPT (0.40) KDM4EALDH1A1ALPLHSD17B10PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009055437-A9 (1,4-DIAZA-BICYCLO[3.2.2]NON-6-EN-4-YL)-HETEROCYCLYL-METHANONE LIGANDS FOR NICOTINIC ACETYLCHOLINE RECEPTORS, USEFUL FOR THE TREATMENT OF DISEASE MEMORY PHARM CORP (US) 2009-07-23 WO disclosed
WO-2009055437-A2 (1,4-DIAZA-BICYCLO[3.2.2]NON-6-EN-4-YL)-HETEROCYCLYL-METHANONE LIGANDS FOR NICOTINIC ACETYLCHOLINE RECEPTORS, USEFUL FOR THE TREATMENT OF DISEASE MEMORY PHARMACEUTICALS CORPORATION (US) 2009-04-30 WO disclosed