SCHEMBL1379181

SCHEMBL1379181

COc1cccc(C(Cc2cccc(NC(=O)CO)n2)(c2cccnc2)c2cccnc2)n1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGER2 P43116 7/20 0.36
GRM5 P41594 3/20 0.35
SORT1 Q99523 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1379534 0.89 PTGER2 (0.36) PTGER2GRM5SORT1
SCHEMBL1381518 0.83 KCNA5 (0.37) PTGER2
SCHEMBL1381052 0.81 GRM5 (0.42) GRM5NPC1RAB9A
SCHEMBL1379427 0.81 NPSR1 (0.47) ADORA3ADORA2A
SCHEMBL3812287 0.80 CYP19A1 (0.33) ADORA3ADORA2A
SCHEMBL3814663 0.79 BACE1 (0.33) ADORA3ADORA2A
SCHEMBL3813507 0.79 NAMPT (0.42) PTGER2GRM5RAB9A
SCHEMBL1382291 0.77 NPC1 (0.37) PTGER2GRM5NPC1RAB9AADORA2A
SCHEMBL3816707 0.76 PTGS2 (0.32)
SCHEMBL1377228 0.75 CYP1A2 (0.43) PTGER2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4719744-B2 2011-07-06 JP claimed
EP-1776355-A4 POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2009-08-12 EP claimed
EP-1776355-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2007-04-25 EP claimed
WO-2006014877-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO claimed