SCHEMBL13801622

SCHEMBL13801622

CC(C)(C)OC(=O)N1CCC(NC(=O)c2cc(Br)cc(C(F)(F)F)c2)[C@H](c2ccc(Br)cc2)C1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.47
USP30 Q70CQ3 6/20 0.45
STS P08842 1/20 0.44
HDAC4 P56524 3/20 0.42
HDAC6 Q9UBN7 2/20 0.42
RORC P51449 1/20 0.41
P2RY14 Q15391 1/20 0.40
FPR2 P25090 3/20 0.40
FPR3 P25089 1/20 0.40
PDE4B Q07343 1/20 0.39
NOTUM Q6P988 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13814606 1.00 TACR1 (0.47) TACR1USP30STSHDAC4HDAC6
SCHEMBL13814605 0.96 TACR1 (0.50) TACR1USP30STSHDAC4HDAC6
SCHEMBL13801621 0.96 TACR1 (0.50) TACR1USP30STSHDAC4HDAC6
SCHEMBL13814602 0.95 TACR1 (0.46) TACR1USP30STSHDAC4HDAC6
SCHEMBL13801602 0.95 TACR1 (0.46) TACR1USP30STSHDAC4HDAC6
SCHEMBL13801594 0.95 TACR1 (0.46) TACR1USP30STSHDAC4HDAC6
SCHEMBL13814677 0.95 TACR1 (0.46) TACR1USP30STSHDAC4HDAC6
SCHEMBL13814651 0.94 TACR1 (0.45) TACR1USP30STSHDAC4HDAC6
SCHEMBL13801604 0.94 TACR1 (0.45) TACR1USP30STSHDAC4HDAC6
SCHEMBL13801632 0.94 TACR1 (0.54) TACR1USP30STSRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8470816-B2 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-06-25 US disclosed
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof NTSR2, NTSR1, HNMT TACR1 9/4885USP30 3991/4885STS 648/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.