SCHEMBL13801647

SCHEMBL13801647

CN(C(=O)C(F)(F)F)[C@@H]1CCNC[C@H]1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.44
SLC6A2 P23975 8/20 0.44
SLC6A4 P31645 6/20 0.44
SLC6A3 Q01959 5/20 0.44
SSTR1 P30872 2/20 0.43
SSTR4 P31391 2/20 0.43
TACR2 P21452 4/20 0.42
TAC3 Q9UHF0 1/20 0.42
KCNH2 Q12809 3/20 0.41
CYP2D6 P10635 1/20 0.41
TACR3 P29371 1/20 0.41
AKT1 P31749 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4144176 0.99 SLC6A2 (0.45) TACR1SLC6A2SLC6A4SLC6A3SSTR1
Hydrochloric Acid SCHEMBL4144170 0.99 SLC6A2 (0.45) TACR1SLC6A2SLC6A4SLC6A3SSTR1
SCHEMBL4153751 0.83 TACR2 (0.61) TACR1SLC6A2SLC6A4SLC6A3TACR2
Hydrochloric Acid SCHEMBL4141232 0.82 TACR1 (0.60) TACR1SLC6A2SLC6A4SLC6A3TACR2
Hydrochloric Acid SCHEMBL4141228 0.82 TACR1 (0.60) TACR1SLC6A2SLC6A4SLC6A3TACR2
Hydrochloric Acid SCHEMBL4141381 0.82 TACR2 (0.60) TACR1SLC6A2SLC6A4SLC6A3TACR2
Hydrochloric Acid SCHEMBL4149798 0.82 TACR1 (0.60) TACR1SLC6A2SLC6A4SLC6A3TACR2
Hydrochloric Acid SCHEMBL4149374 0.82 TACR1 (0.60) TACR1SLC6A2SLC6A4SLC6A3TACR2
SCHEMBL4144959 0.81 TACR2 (0.49) TACR1SLC6A2SLC6A4SLC6A3TACR2
SCHEMBL4144966 0.81 TACR2 (0.49) TACR1SLC6A2SLC6A4SLC6A3TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8470816-B2 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-06-25 US disclosed
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-06-18 US disclosed
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof NTSR2, NTSR1, HNMT TACR1 9/4885SLC6A2 241/4885SLC6A4 271/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.