SCHEMBL13804350

SCHEMBL13804350

CCc1cc(Cl)c(NC)c(C(F)(F)F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.36
HSPA5 P11021 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
LMNA P02545 2/20 0.33
PYCR1 P32322 1/20 0.33
AR P10275 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.33
HTR2A P28223 6/20 0.32
HTR2C P28335 5/20 0.32
HTR2B P41595 5/20 0.32
CYP3A4 P08684 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
S1PR1 P21453 1/20 0.30
SLC6A4 P31645 1/20 0.30
KCNH2 Q12809 1/20 0.30
P2RX7 Q99572 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22155162 0.77 IDO1 (0.39) IDO1HSPA5SIGMAR1LMNAPYCR1
SCHEMBL20669921 0.77 HTR2A (0.30) HTR2AHTR2CSLC6A4KCNH2
SCHEMBL14044235 0.74 RAPGEF4 (0.33) RAPGEF4MEN1KMT2A
SCHEMBL13210657 0.72 ADRB2 (0.38) RAPGEF4HTR2AHTR2CHTR2BKMT2A
SCHEMBL257057 0.71 DAO (0.48) IDO1SIGMAR1LMNAPYCR1FFAR4
SCHEMBL257060 0.71 IDO1 (0.61) IDO1LMNAPYCR1RAPGEF4S1PR1
SCHEMBL22379946 0.70 HSPA5 (0.53) HSPA5LMNACYP3A4MEN1ALDH1A1
SCHEMBL5251032 0.69 HSPA5 (0.38) IDO1HSPA5SIGMAR1PYCR1AR
SCHEMBL10618084 0.67 HTR2A (0.33) SIGMAR1HTR2AHTR2CHTR2BCYP3A4
SCHEMBL1768628 0.67 PDE2A (0.40) RAPGEF4CYP3A4ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547694-B2 Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-16 US disclosed