SCHEMBL13812866

SCHEMBL13812866

CC(C)c1nc(N2CCCCS2(=O)=O)c2cccnc2c1O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALCA P06881 7/20 0.61
COMT P21964 4/20 0.39
KDM4E B2RXH2 4/20 0.35
TP53 P04637 3/20 0.35
ALOX15 P16050 3/20 0.35
HTT P42858 3/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
ALOX12 P18054 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
USP2 O75604 1/20 0.35
IDO1 P14902 1/20 0.35
NPC1 O15118 2/20 0.35
METAP2 P50579 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
HSP90AA1 P07900 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769028 0.83 CALCA (0.74) CALCACOMTKDM4ETP53ALOX15
SCHEMBL4067964 0.82 CALCA (0.69) CALCACOMTKDM4ETP53ALOX15
SCHEMBL4072599 0.81 CALCA (0.68) CALCACOMTKDM4ETP53ALOX15
SCHEMBL966418 0.80 CALCA (0.59) CALCACOMTKDM4ETP53ALOX15
SCHEMBL14435145 0.80 CALCA (0.59) CALCACOMTKDM4ETP53ALOX15
SCHEMBL968119 0.80 CALCA (0.78) CALCACOMTTP53ALOX15NPC1
SCHEMBL7258795 0.80 CALCA (0.69) CALCACOMTKDM4EL3MBTL1RAB9A
SCHEMBL4067727 0.79 CALCA (0.65) CALCACOMTKDM4ETP53ALOX15
SCHEMBL1198641 0.74 CALCA (1.00) CALCASMN1; SMN2
SCHEMBL29393055 0.74 CALCA (1.00) CALCASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664046-B1 AZA-QUINOLINOL PHOSPHONATE INTEGRASE INHIBITOR COMPOUNDS GILEAD SCIENCES INC (US) 2009-06-17 EP disclosed