SCHEMBL13812906

SCHEMBL13812906

Cc1nc(C(=O)NC2CCc3cc(F)ccc32)c(O)c2ncccc12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR2 O60603 1/20 0.45
ADORA2A P29274 2/20 0.44
TRPV1 Q8NER1 5/20 0.43
PDE10A Q9Y233 2/20 0.42
BDKRB1 P46663 1/20 0.40
CALCA P06881 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
RIPK1 Q13546 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13993853 0.90 TRPV1 (0.42) TLR2ADORA2ATRPV1PDE10ACALCA
SCHEMBL13812898 0.77 CALCA (0.41) TLR2CALCAALDH1A1LMNAL3MBTL1
SCHEMBL4071013 0.75 ADORA2A (0.50) ADORA2ATAS1R3TAS1R1TAS1R2RIPK1
SCHEMBL13993858 0.74 CALCA (0.62) ADORA2ACALCA
SCHEMBL17768922 0.74 ADORA2A (0.43) ADORA2ATRPV1PDE10A
SCHEMBL6504246 0.72 CALCA (0.60) CALCA
SCHEMBL4060243 0.71 TAS1R3 (0.49) ADORA2ATAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL4066910 0.71 TAS1R3 (0.49) ADORA2ATAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL599644 0.69 CA12 (0.63) TRPV1PDE10ATAS1R3TAS1R1TAS1R2
SCHEMBL31452698 0.67 PDE10A (0.56) TRPV1PDE10ATAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664046-B1 AZA-QUINOLINOL PHOSPHONATE INTEGRASE INHIBITOR COMPOUNDS GILEAD SCIENCES INC (US) 2009-06-17 EP disclosed