SCHEMBL13817837

SCHEMBL13817837

CC1(C)CC(O)=C(c2ccc(Br)cc2Cl)C(=O)N1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BUB1 O43683 1/20 0.36
HTT P42858 3/20 0.35
TDP2 O95551 1/20 0.35
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HPGD P15428 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
GFER P55789 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PLK4 O00444 1/20 0.33
PLK1 P53350 1/20 0.33
PARP10 Q53GL7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13817835 0.86 HTT (0.43) BUB1HTTALDH1A1SMN1; SMN2HPGD
SCHEMBL13817830 0.83 HTT (0.42) BUB1HTTTDP2ALDH1A1SMN1; SMN2
SCHEMBL13817838 0.78 NCEH1 (0.38) TDP2ALDH1A1SMN1; SMN2CYP1A2KDM4E
SCHEMBL13817791 0.78 HTT (0.38) BUB1HTTALDH1A1HPGDKDM4E
SCHEMBL13817808 0.76 BUB1 (0.32) BUB1HTT
SCHEMBL13817822 0.75 ALDH1A1 (0.40) BUB1HTTALDH1A1HPGDKDM4E
SCHEMBL30512977 0.71 HTT (0.58) HTTTDP2ALDH1A1SMN1; SMN2HPGD
SCHEMBL2355632 0.71 ACACB (0.59) BUB1HTTTDP2HPGDGFER
SCHEMBL13817801 0.70 HTT (0.40) BUB1HTTALDH1A1HPGDKDM4E
SCHEMBL14001512 0.68 GSK3B (0.44) HTTALDH1A1SMN1; SMN2HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547660-B2 Phenyl-substituted 4-hydroxy-tetrahydropyridones BAYER AKTIENGESELLSCHAFT (DE) 2009-06-16 US disclosed
US-7547660-B2 Phenyl-substituted 4-hydroxy-tetrahydropyridones BAYER AKTIENGESELLSCHAFT (DE) 2009-06-16 US disclosed