SCHEMBL13819201

SCHEMBL13819201

Bc1c[nH]c(=O)c2c1[nH]c1ccc(F)cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 1/20 0.49
CDK5R1 Q15078 1/20 0.49
FEN1 P39748 1/20 0.43
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 2/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
JAK2 O60674 1/20 0.40
CDC25A P30304 1/20 0.40
CDC25C P30307 1/20 0.40
PGR P06401 2/20 0.39
DAO P14920 1/20 0.39
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
MPO P05164 1/20 0.38
CDK4 P11802 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13819449 0.82 CDK5 (0.43) CDK5CDK5R1FEN1KDM4EALDH1A1
SCHEMBL3508562 0.82 CDK5 (0.43) CDK5CDK5R1FEN1KDM4EALDH1A1
SCHEMBL3506366 0.79 CLK1 (0.50) CDK5CDK5R1FEN1KDM4EALDH1A1
SCHEMBL5879244 0.73 CHEK1 (0.59) CDK5CDK5R1FEN1KDM4EALDH1A1
SCHEMBL797858 0.72 KDM4E (0.50) FEN1KDM4EALDH1A1GLAGAA
SCHEMBL3251991 0.70 KDM4E (0.58) CDK5CDK5R1FEN1KDM4EALDH1A1
SCHEMBL13417447 0.70 KDM4E (0.65) CDK5CDK5R1FEN1KDM4EALDH1A1
SCHEMBL22566960 0.69 CDK4 (0.71) CDK5CDK5R1CDK4CCND1CCNE2
SCHEMBL5821446 0.68 ROCK2 (0.52) CDK5CDK5R1
SCHEMBL17613784 0.66 CDK5 (0.47) CDK5CDK5R1FEN1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009075830-A1 INHIBITORS OF JANUS KINASES MERCK & CO., INC. (US) 2009-06-18 WO disclosed