SCHEMBL13819984

SCHEMBL13819984

Cc1ccc(Cn2cc(CNC(=O)c3coc(-c4ccccc4)n3)nn2)cc1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.54
KLKB1 P03952 3/20 0.49
KDM5B Q9UGL1 2/20 0.48
HDAC1 Q13547 4/20 0.47
HDAC8 Q9BY41 3/20 0.47
HDAC6 Q9UBN7 3/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SCD O00767 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12339960 0.95 HDAC1 (0.52) MAOBKLKB1KDM5BHDAC1HDAC8
SCHEMBL12339937 0.93 HDAC1 (0.50) MAOBKLKB1KDM5BHDAC1HDAC8
SCHEMBL12339963 0.86 TUBB4A (0.57) MAOBKLKB1KDM5B
SCHEMBL12339950 0.85 HDAC1 (0.49) MAOBKLKB1HDAC1HDAC8HDAC6
SCHEMBL12902828 0.85 MAOB (0.48) MAOBKLKB1HDAC1HDAC8HDAC6
SCHEMBL12339928 0.83 TUBB4A (0.54) MAOBKLKB1KDM5B
SCHEMBL13819976 0.83 ANPEP (0.54) HDAC1HDAC8HDAC6
SCHEMBL12339961 0.81 TUBB4A (0.44) MAOBKDM5BHDAC1HDAC8HDAC6
SCHEMBL12339962 0.80 HDAC1 (0.48) HDAC1HDAC8HDAC6
SCHEMBL12339959 0.80 TUBB4A (0.51) MAOBKLKB1KDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8729270-B2 Anti-cancer compounds, synthesis thereof, and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2014-05-20 US disclosed
US-8729270-B2 Anti-cancer compounds, synthesis thereof, and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2014-05-20 US disclosed
US-20120289704-A1 ANTI-CANCER COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2012-11-15 US disclosed
US-20120289704-A1 ANTI-CANCER COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2012-11-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120289704-A1 ANTI-CANCER COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME MCL1, BRDT, GLS MAOB 1529/4885KLKB1 2046/4885KDM5B 551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.