SCHEMBL13823906

SCHEMBL13823906

C[C@@]1(c2ccc(-c3cccnc3)cc2)C(=O)N(c2cc(Cl)cc(Cl)c2)c2nccn21

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 5/20 0.48
ICAM1 P05362 5/20 0.48
ITGAL P20701 5/20 0.48
MCHR1 Q99705 4/20 0.39
MAPKAPK2 P49137 1/20 0.37
BACE1 P56817 5/20 0.36
CTSD P07339 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
PSD A5PKW4 1/20 0.36
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13817292 0.84 ITGB2 (0.70) ITGB2ICAM1ITGAL
SCHEMBL13823838 0.79 ITGAL (0.51) ITGB2ICAM1ITGAL
SCHEMBL13817170 0.74 ITGB2 (0.77) ITGB2ICAM1ITGAL
SCHEMBL4238659 0.73 ITGB2 (0.72) ITGB2ICAM1ITGAL
SCHEMBL13816995 0.70 ITGB2 (0.73) ITGB2ICAM1ITGAL
SCHEMBL13817154 0.68 ITGB2 (0.79) ITGB2ICAM1ITGAL
SCHEMBL7672836 0.65 MCHR1 (0.38) ITGB2ICAM1ITGALMCHR1CYP11B1
SCHEMBL14019343 0.65 ITGB2 (0.81) ITGB2ICAM1ITGAL
SCHEMBL13817322 0.65 ITGB2 (0.80) ITGB2ICAM1ITGAL
SCHEMBL4018223 0.65 ITGB2 (1.00) ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7550494-B2 Small molecules useful in the treatment of inflammatory disease BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2009-06-23 US disclosed