SCHEMBL7672836

SCHEMBL7672836

C[C@@]12C(=O)N(c3cc(Cl)cc(Cl)c3)C(=O)N1CC[C@@H]2c1ccc(-c2cccnc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.38
CYP3A4 P08684 1/20 0.37
ITGAL P20701 5/20 0.36
CYP11B1 P15538 2/20 0.36
CYP17A1 P05093 1/20 0.36
CYP21A2 P08686 1/20 0.36
FPR1 P21462 1/20 0.36
FPR2 P25090 1/20 0.36
CYP11B2 P19099 1/20 0.35
APP P05067 1/20 0.35
GRM2 Q14416 1/20 0.35
LMNA P02545 1/20 0.35
ITGB2 P05107 1/20 0.35
ICAM1 P05362 1/20 0.35
CCR1 P32246 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7665393 0.82 ITGAL (0.41) ITGALITGB2ICAM1
SCHEMBL7665397 0.82 ITGAL (0.41) ITGALITGB2ICAM1
SCHEMBL7663043 0.80 ITGAL (0.46) ITGALITGB2ICAM1
SCHEMBL4848485 0.70 MCHR1 (0.40) MCHR1CYP3A4ITGALCYP11B1CYP11B2
SCHEMBL14526280 0.66 GRM2 (0.38) MCHR1CYP3A4ITGALCYP11B1CYP11B2
SCHEMBL3839434 0.65 ITGAL (0.52) ITGALITGB2ICAM1
SCHEMBL3839432 0.65 ITGAL (0.52) ITGALITGB2ICAM1
SCHEMBL13823906 0.65 ITGB2 (0.48) MCHR1ITGALCYP11B1CYP11B2ITGB2
SCHEMBL13817292 0.64 ITGB2 (0.70) ITGALITGB2ICAM1
SCHEMBL3838174 0.64 ITGAL (0.68) ITGALITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365615-B1 DICHLOROPHENYL TETRAHYDROPYRROLO(1,2-C)IMIDAZOLE-1,3-DIONES; IMMUNE CELL MEDIATED CONDITIONS; ANTAGONISTS OF THE BINDING OF HUMON INTERCELLULAR ADHESION MOLECULES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-04-02 US claimed
WO-2001007052-A1 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-02-01 WO claimed
US-6365615-B1 DICHLOROPHENYL TETRAHYDROPYRROLO(1,2-C)IMIDAZOLE-1,3-DIONES; IMMUNE CELL MEDIATED CONDITIONS; ANTAGONISTS OF THE BINDING OF HUMON INTERCELLULAR ADHESION MOLECULES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-04-02 US disclosed