SCHEMBL13832504

SCHEMBL13832504

COc1cc(F)c(N)cc1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.52
POLB P06746 1/20 0.52
GAA P10253 2/20 0.50
ALDH1A1 P00352 7/20 0.46
CYP3A4 P08684 3/20 0.46
TDP1 Q9NUW8 3/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
PKM P14618 1/20 0.44
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
KMT2A Q03164 1/20 0.43
S100B P04271 1/20 0.42
NPC1 O15118 1/20 0.40
HTT P42858 2/20 0.39
LMNA P02545 1/20 0.39
ADRA2B P18089 1/20 0.39
PTGS1 P23219 1/20 0.39
KIT P10721 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1766204 0.88 NPC1 (0.46) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL30313255 0.88 L3MBTL1 (0.54) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL569225 0.88 L3MBTL1 (0.54) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL19385593 0.86 L3MBTL1 (0.52) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL30661038 0.86 ALDH1A1 (0.41) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL13195018 0.86 ALDH1A1 (0.41) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL14566064 0.82 TAAR1 (0.46) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL5466626 0.82 L3MBTL1 (0.48) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL453951 0.82 GAA (0.68) L3MBTL1POLBGAAALDH1A1CYP3A4
SCHEMBL1708520 0.81 NPC1 (0.45) L3MBTL1POLBGAAALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181217-B Pyrazolo [1,5-a ] [1,3,5] triazine derivative and salt thereof and application of derivative and salt thereof in preparation of anti-cancer drugs 陕西师范大学 2022-12-27 CN disclosed
CN-114181217-A Pyrazolo [1,5-a ] [1,3,5] triazine derivative and salt thereof and application of derivative and salt thereof in preparation of anti-cancer drugs 陕西师范大学 2022-03-15 CN disclosed
EP-3885344-A2 PYRIMIDINE COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USES THEREOF InventisBio Co., Ltd. (CN) 2021-09-29 EP disclosed
EP-2844642-B1 COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS ARIAD PHARMA INC (US) 2019-11-13 EP disclosed
CN-106458969-A (substituted phenyl) (substituted pyrimidine) amino derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2017-02-22 CN disclosed
WO-2012151561-A1 COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS ARIAD PHARMACEUTICALS, INC. (US) 2012-11-08 WO disclosed