SCHEMBL138377

SCHEMBL138377

O=S(=O)(NCc1ccccc1C(F)(F)F)C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.46
CA2 P00918 1/20 0.45
NAMPT P43490 1/20 0.44
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
EPHX2 P34913 2/20 0.43
RECQL P46063 1/20 0.43
IDO1 P14902 2/20 0.43
LMNA P02545 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
KMT2A Q03164 1/20 0.42
HPGD P15428 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30810439 0.83 NPSR1 (0.52) NPSR1NAMPTKDM4EALDH1A1TDP1
SCHEMBL138368 0.81 LMNA (0.68) NPSR1CA2KDM4ERECQLLMNA
SCHEMBL30927226 0.80 NAMPT (0.56) CA2NAMPTKDM4EALDH1A1TDP1
SCHEMBL140452 0.79 MEN1 (0.55) CA2ALDH1A1LMNAKMT2AHPGD
SCHEMBL139590 0.79 HPGD (0.51) CA2LMNAKMT2AHPGD
SCHEMBL140457 0.79 PTGS1 (0.50) CA2ALDH1A1LMNAKMT2AHPGD
SCHEMBL21679846 0.77 IDO1 (0.52) NPSR1KDM4EALDH1A1TDP1EPHX2
SCHEMBL17201441 0.77 CA2 (0.55) CA2LMNA
SCHEMBL20906520 0.77 CA2 (0.64) CA2TDP1LMNAKMT2AHPGD
SCHEMBL138386 0.76 CA2 (0.42) CA2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120059179-A1 PALLADIUM-CATALYZED ORTHO-FLUORINATION The Scripps Research Insitiute (US) 2012-03-08 US disclosed
WO-2010115098-A2 PALLADIUM-CATALYZED ORTHO-FLUORINATION THE SCRIPPS RESEARCH INSTITUTE (US) 2010-10-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059179-A1 PALLADIUM-CATALYZED ORTHO-FLUORINATION POF1B, OCIAD2, ODC1 NPSR1 1553/4885CA2 3314/4885NAMPT 1358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.