SCHEMBL1384364

SCHEMBL1384364

Cc1c(C(N)=O)ccn1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
KDM6A O15550 1/20 0.45
KDM4A O75164 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KDM5C P41229 1/20 0.45
KDM2B Q8NHM5 1/20 0.45
DOHH Q9BU89 1/20 0.45
KDM2A Q9Y2K7 1/20 0.45
SIRT3 Q9NTG7 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NOTUM Q6P988 2/20 0.36
MAPT P10636 3/20 0.35
HPGD P15428 2/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HSD17B10 Q99714 1/20 0.35
NNMT P40261 1/20 0.35
PARP1 P09874 2/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4562515 0.80 NOTUM (0.55) KDM4EKDM6AKDM4ACYP2C9CYP2C19
SCHEMBL16217227 0.79 KDM4E (0.42) KDM4EKDM6AKDM4ACYP2C9CYP2C19
SCHEMBL25072434 0.78 KDM4E (0.35) KDM4EKDM6AKDM4ACYP2C9CYP2C19
Hydrochloric Acid SCHEMBL30678145 0.78 NOTUM (0.53) KDM4EKDM6AKDM4ACYP2C9CYP2C19
SCHEMBL28202433 0.78 SIRT3 (0.38) KDM4ESIRT3TDP1NOTUMMAPT
SCHEMBL19651995 0.78 SIRT3 (0.39) KDM4EKDM6AKDM4ACYP2C9CYP2C19
SCHEMBL9736660 0.77 CYP2C19 (0.44) KDM4EKDM6AKDM4ACYP2C9CYP2C19
SCHEMBL16418351 0.75 KDM4E (0.46) KDM4EKDM6AKDM4ACYP2C9CYP2C19
SCHEMBL16417043 0.75 BRD4 (0.45) KDM4EKDM6AKDM4ACYP2C9CYP2C19
SCHEMBL31748394 0.74 KDM4E (0.55) KDM4EKDM6AKDM4ACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109320499-A Pyrrole-3-carboxamide class compound and its preparation method and application 沈阳药科大学 2019-02-12 CN claimed
JP-4703649-B2 2011-06-15 JP claimed
EP-1773768-A4 PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS EXELIXIS INC (US) 2008-08-06 EP claimed
EP-1773768-A2 PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS Exelixis, Inc. (US) 2007-04-18 EP claimed
WO-2006012642-A2 PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS EXELIXIS, INC. (US) 2006-02-02 WO claimed
WO-2025233641-A1 NOVEL PHOTOINDUCIBLE KINASE INHIBITORS FOR TREATING PROLIFERATIVE AND VASOPROLIFERATIVE DISEASES SEMMELWEIS EGYETEM (HU) 2025-11-13 WO disclosed
US-20250115577-A1 BCL-2 Inhibitors Eil Therapeutics, Inc. 2025-04-10 US disclosed
CN-119053587-A 5- [7- (3, 4-Dihydro-1H-isoquinoline-2-carbonyl) -1,2,3,4 tetrahydroisoquinolin-6-yl ] -1H-pyrrole-3-carboxamide derivatives, pharmaceutical compositions containing same and use thereof as pro-apoptotic agents 法国施维雅药厂 2024-11-29 CN disclosed
EP-4457223-A1 BCL-2 INHIBITORS Eil Therapeutics, Inc. (US) 2024-11-06 EP disclosed
CN-118451070-A BCL-2 inhibitors 伊尔治疗学股份有限公司 2024-08-06 CN disclosed
US-12053465-B2 KCC2 expression enhancing compounds and uses thereof WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2024-08-06 US disclosed
WO-2023129553-A1 BCL-2 INHIBITORS Eil Therapeutics, Inc. (US) 2023-07-06 WO disclosed
CN-109456324-B Isoindoline or isoquinoline compounds, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2022-04-22 CN disclosed
US-20200085817-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2020-03-19 US disclosed
CN-105408320-B 3- (aryl or heteroaryl) methyl indol -2- ketone derivatives as cancer stem cell approach kinase inhibitor for treating cancer 北京强新生物科技有限公司 2019-08-13 CN disclosed
CN-109456324-A New isoindoline or isoquinoline compound, preparation method and the Pharmaceutical composition containing them 法国施维雅药厂 2019-03-12 CN disclosed
CN-109320499-A Pyrrole-3-carboxamide class compound and its preparation method and application 沈阳药科大学 2019-02-12 CN disclosed
WO-2018217766-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2018-11-29 WO disclosed
EP-2970206-A1 3-(ARYL OR HETEROARYL) METHYLENEINDOLIN-2-ONE DERIVATIVES AS INHIBITORS OF CANCER STEM CELL PATHWAY KINASES FOR THE TREATMENT OF CANCER Boston Biomedical, Inc. (US) 2016-01-20 EP disclosed
WO-2014160401-A1 3-(ARYL OR HETEROARYL) METHYLENEINDOLIN-2-ONE DERIVATIVES AS INHIBITORS OF CANCER STEM CELL PATHWAY KINASES FOR THE TREATMENT OF CANCER BOSTON BIOMEDICAL, INC. (US) 2014-10-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200085817-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF MECP2, SLC1A2, GRIN2C KDM4E 127/4885KDM6A 197/4885KDM4A 151/4885
US-20250115577-A1 BCL-2 Inhibitors BCL2, BCL2L1, BCL2L2 KDM4E 3326/4885KDM6A 3166/4885KDM4A 3716/4885
US-12053465-B2 KCC2 expression enhancing compounds and uses thereof MECP2, SLC1A2, GRIN2C KDM4E 127/4885KDM6A 197/4885KDM4A 151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.