SCHEMBL13844166

SCHEMBL13844166

Cc1nnc(-c2cc(N)c(F)cc2F)o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
NOTUM Q6P988 2/20 0.38
LRRK2 Q5S007 3/20 0.36
BRD4 O60885 2/20 0.34
PDK2 Q15119 1/20 0.34
BACE1 P56817 2/20 0.33
TRPM8 Q7Z2W7 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
CASP3 P42574 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
KDM4E B2RXH2 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21939245 0.78 NOTUM (0.43) CA12CA1CA2CA9NOTUM
SCHEMBL13451187 0.75 NOTUM (0.46) NOTUMBACE1NPC1RAB9ASMN1; SMN2
SCHEMBL13103800 0.74 NOTUM (0.42) CA12CA1CA2CA9NOTUM
SCHEMBL16573949 0.74 NOTUM (0.45) CA12CA1CA2CA9NOTUM
SCHEMBL26206906 0.74 NOTUM (0.45) CA12CA1CA2CA9NOTUM
SCHEMBL21958452 0.72 LRRK2 (0.48) CA12CA1CA2CA9NOTUM
SCHEMBL8103862 0.71 NOTUM (0.40) CA12CA1CA2CA9NOTUM
SCHEMBL4287576 0.71 GPR84 (0.40) CA12CA1CA2CA9NOTUM
SCHEMBL1187141 0.71 ESR1 (0.47) NOTUM
SCHEMBL2898396 0.71 NOTUM (0.43) CA12CA1CA2CA9NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009058919-A1 CCR5 ANTAGONISTS AS THERAPEUTIC AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2009-05-07 WO disclosed