SCHEMBL13844901

SCHEMBL13844901

Nc1ccc(S(=O)(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1

nearest known ligand 0.77

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.77
KMT2A Q03164 4/20 0.69
MEN1 O00255 3/20 0.69
POLB P06746 2/20 0.55
EPHX2 P34913 1/20 0.55
HSD11B1 P28845 1/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
NAMPT P43490 1/20 0.53
KDM4E B2RXH2 2/20 0.52
GAA P10253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6211593 0.93 ALDH1A1 (0.87) ALDH1A1KMT2AMEN1POLBEPHX2
SCHEMBL7406370 0.87 ALDH1A1 (1.00) ALDH1A1KMT2AMEN1POLBHSD11B1
SCHEMBL5468343 0.85 ALDH1A1 (0.74) ALDH1A1KMT2AMEN1POLBEPHX2
SCHEMBL5468345 0.85 ALDH1A1 (0.74) ALDH1A1KMT2AMEN1POLBEPHX2
SCHEMBL6210846 0.81 ALDH1A1 (0.71) ALDH1A1KMT2AMEN1POLBEPHX2
SCHEMBL28224185 0.81 ALDH1A1 (0.66) ALDH1A1KMT2AMEN1POLBEPHX2
SCHEMBL2636523 0.79 MAPT (0.70) ALDH1A1KMT2AMEN1POLBEPHX2
SCHEMBL10674722 0.79 CA12 (0.66) ALDH1A1KMT2AMEN1POLBL3MBTL1
SCHEMBL10717731 0.79 CA12 (0.66) ALDH1A1KMT2AMEN1POLBL3MBTL1
SCHEMBL6210077 0.79 HSD11B1 (0.86) ALDH1A1POLBHSD11B1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009056693-A1 NOVEL DERIVATIVES OF N, N'- 2, 4-DIANILINOPYRIMIDINES, PREPARATION THEREOF AS MEDICAMENTS PHARMACEUTICAL COMPOSITIONS AND IN PARTICULAR AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2009-05-07 WO disclosed