SCHEMBL13845164

SCHEMBL13845164

CCOC(=O)c1cccc(-c2cccc(CNc3nc(NC[C@@H]4CCNC4)ncc3N)c2C)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 1/20 0.41
PTGER4 P35408 1/20 0.40
IRAK4 Q9NWZ3 4/20 0.38
IRAK1 P51617 2/20 0.38
TYRO3 Q06418 1/20 0.37
PRKCQ Q04759 4/20 0.36
PIK3CA P42336 1/20 0.36
CHRM3 P20309 2/20 0.36
AURKA O14965 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
BRAF P15056 1/20 0.35
BTK Q06187 1/20 0.35
ITK Q08881 1/20 0.35
DGAT2 Q96PD7 1/20 0.35
PTK2 Q05397 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13978066 0.87 PRKCQ (0.50) PTGER4IRAK1PRKCQCYP3A4CYP2C9
SCHEMBL13608140 0.81 PIK3CA (0.40) ACP1IRAK4IRAK1PIK3CACHRM3
SCHEMBL13845177 0.80 PRKCQ (0.51) IRAK4IRAK1TYRO3PRKCQCYP3A4
SCHEMBL13978067 0.77 PRKCQ (0.45) IRAK1TYRO3PRKCQCYP3A4CYP2C9
SCHEMBL13978061 0.77 PRKCQ (0.58) IRAK1PRKCQCYP3A4CYP2C9
SCHEMBL13845174 0.75 PRKCQ (0.48) IRAK1TYRO3PRKCQCYP3A4CYP2C9
SCHEMBL13608118 0.73 FYN (0.38) ACP1IRAK4IRAK1TYRO3
SCHEMBL13978063 0.73 PRKCQ (0.56) IRAK1PRKCQCYP3A4CYP2C9
SCHEMBL13978062 0.73 PRKCQ (0.46) IRAK1TYRO3PRKCQCYP3A4CYP2C9
SCHEMBL13978291 0.73 ACACB (0.40) PRKCQCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009062059-A2 ISOMERIC PURINONES AND 1H-IMIDAZOPYRIDINONES AS PKC-THETA INHIBITORS PHARMACOPEIA, INC. (US) 2009-05-14 WO disclosed