SCHEMBL13845253

SCHEMBL13845253

Nc1cnc(NC[C@@H]2CCNC2)cc1NCc1cccc(Cl)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 9/20 0.43
PRKCQ Q04759 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
SLC6A2 P23975 4/20 0.38
SLC6A4 P31645 4/20 0.38
SLC6A3 Q01959 4/20 0.38
CYP2D6 P10635 3/20 0.38
KDM1A O60341 1/20 0.38
RPS6KB1 P23443 2/20 0.37
IRAK4 Q9NWZ3 2/20 0.36
IRAK1 P51617 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3845255 0.78 PRKCQ (0.40) CCNT1PRKCQCYP3A4CYP2C9CYP2D6
SCHEMBL3984172 0.75 PRKCQ (0.60) CCNT1PRKCQCYP3A4CYP2C9CYP2D6
SCHEMBL13608022 0.75 CDK9 (0.42) CCNT1PRKCQCYP3A4CYP2C9SLC6A2
SCHEMBL13608017 0.74 CCNT1 (0.45) CCNT1IRAK1
SCHEMBL13846484 0.73 PRKCQ (0.49) CCNT1PRKCQCYP3A4CYP2C9CYP2D6
SCHEMBL3844951 0.69 CD38 (0.44) CYP3A4RPS6KB1
SCHEMBL30137522 0.69 PTPN11 (0.52) CCNT1KDM1A
SCHEMBL13846476 0.67 PRKCQ (0.60) PRKCQCYP3A4CYP2C9CYP2D6IRAK1
SCHEMBL3987070 0.67 PRKCQ (0.70) PRKCQCYP3A4CYP2C9CYP2D6IRAK1
SCHEMBL13845174 0.67 PRKCQ (0.48) PRKCQCYP3A4CYP2C9CYP2D6KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009062059-A2 ISOMERIC PURINONES AND 1H-IMIDAZOPYRIDINONES AS PKC-THETA INHIBITORS PHARMACOPEIA, INC. (US) 2009-05-14 WO disclosed