SCHEMBL13845922

SCHEMBL13845922

COCC(C)(C)C/C=C/c1cccc(I)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.48
CACNA1B Q00975 1/20 0.34
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
IDO1 P14902 2/20 0.33
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
RELA Q04206 1/20 0.31
GRIK1 P39086 1/20 0.31
GRIK2 Q13002 1/20 0.31
MMP1 P03956 1/20 0.30
MMP9 P14780 1/20 0.30
MMP13 P45452 1/20 0.30
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13845999 0.86 APP (0.46) APPCACNA1BCHRM2CHRM1CHRM3
SCHEMBL8000869 0.84 RELA (0.46) CACNA1BCHRM2CHRM1CHRM3IDO1
SCHEMBL13845927 0.74 CYP1A1 (0.35)
SCHEMBL13845994 0.73 APP (0.50) APPCACNA1BCHRM2CHRM1CHRM3
SCHEMBL15050807 0.72 APP (0.52) APPCACNA1BCHRM2CHRM1CHRM3
SCHEMBL15050808 0.72 APP (0.52) APPCACNA1BCHRM2CHRM1CHRM3
SCHEMBL13845988 0.72 APP (0.49) APPCACNA1BCHRM2CHRM1CHRM3
SCHEMBL13846004 0.71 APP (0.46) APPCACNA1BCHRM2CHRM1CHRM3
SCHEMBL13846023 0.71 APP (0.48) APPCACNA1BCHRM2CHRM1CHRM3
SCHEMBL7999307 0.70 RELA (0.44) CHRM2CHRM1CHRM3IDO1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009064955-A1 MACROCYCLIC TETRAZOLYL HEPATITIS C SERINE PROTEASE INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-05-22 WO disclosed