SCHEMBL13845993

SCHEMBL13845993

COc1ccc(I)cc1/C=C/CCCC(C)(C)OC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.35
AR P10275 1/20 0.35
JUN P05412 1/20 0.34
NFKB1 P19838 1/20 0.34
CYP1A1 P04798 3/20 0.33
CYP1B1 Q16678 3/20 0.33
NFE2L2 Q16236 2/20 0.33
CYP1A2 P05177 1/20 0.33
KDM4E B2RXH2 2/20 0.33
KMT2A Q03164 1/20 0.33
MAPT P10636 2/20 0.32
APP P05067 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
CXCL12 P48061 1/20 0.32
CAPN1 P07384 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7991057 0.85 PDE5A (0.40) BACE1JUNNFKB1CYP1A1CYP1B1
SCHEMBL13845981 0.85 BACE1 (0.36) BACE1ARJUNNFKB1CYP1A1
SCHEMBL7990211 0.82 PDE5A (0.37) BACE1CYP1A1CYP1B1NFE2L2CYP1A2
SCHEMBL13845936 0.81 CYP1A1 (0.36) BACE1ARJUNNFKB1CYP1A1
SCHEMBL13845930 0.81 CYP1A1 (0.36) BACE1ARJUNNFKB1CYP1A1
SCHEMBL13845935 0.80 CYP1A1 (0.36) BACE1ARJUNNFKB1CYP1A1
SCHEMBL13845921 0.79 CYP1A1 (0.33) BACE1ARJUNNFKB1CYP1A1
SCHEMBL13846057 0.78 L3MBTL4 (0.43) BACE1ARJUNNFKB1CYP1A1
SCHEMBL13846066 0.77 L3MBTL4 (0.45) BACE1ARCYP1A1CYP1B1NFE2L2
SCHEMBL8002469 0.77 ACHE (0.40) BACE1JUNNFKB1CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009064955-A1 MACROCYCLIC TETRAZOLYL HEPATITIS C SERINE PROTEASE INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-05-22 WO disclosed