SCHEMBL13846100

SCHEMBL13846100

COc1cc(C(=O)NC[C@H]2CCNC2)ccc1N

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 2/20 0.61
SMYD3 Q9H7B4 3/20 0.55
NAMPT P43490 3/20 0.50
ROCK2 O75116 4/20 0.49
TDP1 Q9NUW8 1/20 0.49
PKN2 Q16513 1/20 0.48
BRD4 O60885 1/20 0.48
MAPK14 Q16539 1/20 0.47
F10 P00742 1/20 0.45
TOP2A P11388 2/20 0.44
ROCK1 Q13464 1/20 0.44
CHEK2 O96017 1/20 0.44
MET P08581 1/20 0.44
SUV39H2 Q9H5I1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13575608 1.00 HTR4 (0.61) HTR4SMYD3NAMPTROCK2TDP1
SCHEMBL13846092 1.00 HTR4 (0.61) HTR4SMYD3NAMPTROCK2TDP1
SCHEMBL13846145 0.93 HTR4 (0.59) HTR4SMYD3ROCK2TDP1PKN2
SCHEMBL13846148 0.93 HTR4 (0.59) HTR4SMYD3ROCK2TDP1PKN2
SCHEMBL13846080 0.93 HTR4 (0.67) HTR4SMYD3ROCK2TDP1BRD4
SCHEMBL4802575 0.88 HTR4 (0.72) HTR4ROCK2TDP1MAPK14F10
SCHEMBL13175546 0.85 HTR4 (0.69) HTR4TDP1MAPK14F10
SCHEMBL13175812 0.85 HTR4 (0.69) HTR4ROCK2TDP1MAPK14F10
SCHEMBL13175544 0.84 TDP1 (0.69) HTR4TDP1MAPK14
SCHEMBL13175541 0.82 HTR4 (0.66) HTR4NAMPTROCK2TDP1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009067547-A1 POLO-LIKE KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-05-28 WO disclosed