SCHEMBL13848745

SCHEMBL13848745

CCOC(=O)Cc1nc(N)c(C#N)c(-c2ccc3c(c2)OCCO3)c1C#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.52
ADORA2A P29274 1/20 0.52
ALDH1A1 P00352 11/20 0.47
KDM4E B2RXH2 10/20 0.47
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
RECQL P46063 1/20 0.47
HIF1A Q16665 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 7/20 0.46
HPGD P15428 6/20 0.46
MAPT P10636 6/20 0.46
HSD17B10 Q99714 4/20 0.46
RXFP1 Q9HBX9 3/20 0.46
GAA P10253 3/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
TSHR P16473 4/20 0.44
LMNA P02545 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13848718 0.94 ADORA1 (0.59) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL5951009 0.86 ADORA1 (0.53) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL4191367 0.82 ADORA1 (0.51) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL5951208 0.77 ADORA1 (0.57) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL4022211 0.76 ADORA1 (0.58) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL4030275 0.74 ADORA1 (0.53) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL3342911 0.73 ADORA1 (0.59) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL3548181 0.73 ADORA1 (0.62) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL4024284 0.73 ADORA1 (0.58) ADORA1ADORA2AALDH1A1KDM4EMEN1
SCHEMBL3554077 0.72 ADORA1 (0.78) ADORA1ADORA2AALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377570-B1 SUBSTITUTED 2-CARBA-3,5-DICYANO-4-ARYL-6-AMINOPYRIDINES AND THE USE OF THE SAME AS SELECTIVE LIGANDS OF THE ADENOSINE RECEPTOR BAYER HEALTHCARE AG (DE) 2009-05-13 EP disclosed