SCHEMBL13849641

SCHEMBL13849641

C=C1NN=C(c2ccc3c(c2)nc(-c2ccc(OC)cc2)n3Cc2ccccc2)C(C)S1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.57
HTT P42858 7/20 0.57
MAPT P10636 6/20 0.57
SMN1; SMN2 Q16637 5/20 0.57
TP53 P04637 5/20 0.57
HPGD P15428 5/20 0.57
NPSR1 Q6W5P4 2/20 0.57
KDM4E B2RXH2 6/20 0.53
LMNA P02545 2/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
CNR2 P34972 1/20 0.53
BRD4 O60885 4/20 0.49
GAA P10253 2/20 0.47
POLB P06746 1/20 0.45
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 P62805 1/20 0.43
PDE6D O43924 2/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3617954 0.90 ALDH1A1 (0.57) ALDH1A1HTTMAPTSMN1; SMN2TP53
SCHEMBL5582025 0.71 ALDH1A1 (1.00) ALDH1A1HTTMAPTSMN1; SMN2TP53
SCHEMBL30789276 0.70 TP53 (0.71) ALDH1A1HTTMAPTSMN1; SMN2TP53
SCHEMBL10443668 0.70 ALDH1A1 (0.92) ALDH1A1HTTMAPTSMN1; SMN2TP53
SCHEMBL29974892 0.69 PDE3B (0.59) ALDH1A1HTTMAPTSMN1; SMN2TP53
SCHEMBL3440842 0.69 MEN1 (0.43) ALDH1A1SMN1; SMN2BRD4MEN1KMT2A
SCHEMBL6475362 0.69 ALDH1A1 (0.74) ALDH1A1HTTMAPTSMN1; SMN2TP53
SCHEMBL10443667 0.69 ALDH1A1 (0.82) ALDH1A1HTTMAPTSMN1; SMN2TP53
SCHEMBL3440841 0.68 PTGER4 (0.47) BRD4
SCHEMBL8024196 0.68 TP53 (0.62) ALDH1A1HTTMAPTSMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058308-A1 Benzimidazoledihydrothiadiazinone derivatives used as fructose-1,6-biphosphatase inhibitors and pharmaceutical compositions containing same. Merck Sante (FR) 2009-05-13 EP disclosed