SCHEMBL1385162

SCHEMBL1385162

O=C(Nc1cccc(Cl)c1)c1nccnc1Nc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 2/20 0.61
HDAC6 Q9UBN7 1/20 0.60
NPC1 O15118 4/20 0.57
RAB9A P51151 4/20 0.57
KDR P35968 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.53
HIF1A Q16665 1/20 0.53
MAPT P10636 3/20 0.53
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
LMNA P02545 1/20 0.52
HTT P42858 1/20 0.52
KCNK3 O14649 1/20 0.51
KCNK9 Q9NPC2 1/20 0.51
AHR P35869 1/20 0.51
FADS1 O60427 1/20 0.50
P4HTM Q9NXG6 1/20 0.50
POLB P06746 1/20 0.50
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1386612 0.88 GRM4 (0.59) GRM4HDAC6NPC1RAB9AKDR
SCHEMBL28501806 0.82 GRM4 (0.68) GRM4HDAC6NPC1RAB9AKDR
SCHEMBL29516188 0.82 GRM4 (0.68) GRM4HDAC6NPC1RAB9AKDR
SCHEMBL1383789 0.81 GRM5 (0.51) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL17685484 0.79 MAPT (0.51) GRM4HDAC6NPC1RAB9AKDR
SCHEMBL14284353 0.77 GRM4 (0.73) GRM4HDAC6NPC1RAB9AKDR
SCHEMBL29496401 0.76 GRM4 (1.00) GRM4HDAC6NPC1RAB9AKDR
SCHEMBL2530324 0.76 GRM4 (1.00) GRM4HDAC6NPC1RAB9AKDR
SCHEMBL16007573 0.76 KDR (0.70) GRM4HDAC6RAB9AKDRSMN1; SMN2
SCHEMBL4134533 0.75 DHODH (0.62) NPC1RAB9ASMN1; SMN2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4774410-B2 2011-09-14 JP claimed
US-7947685-B2 Pyrazine-2-carboxyamide derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-24 US disclosed