SCHEMBL13857005

SCHEMBL13857005

COc1cc(F)c2nccc(NC(=O)N3CCC(NCc4cc5c(F)ccc(F)c5[nH]4)CC3)c2c1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 9/20 0.55
NOS3 P29474 3/20 0.37
NOS1 P29475 3/20 0.37
NOS2 P35228 3/20 0.37
S1PR2 O95136 1/20 0.36
KCNH2 Q12809 2/20 0.36
PAK1 Q13153 2/20 0.35
ERBB2 P04626 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5773953 0.89 SLC2A1 (0.53) SLC2A1NOS3NOS1NOS2KCNH2
SCHEMBL13857009 0.83 SLC2A1 (0.65) SLC2A1KCNH2
SCHEMBL4270077 0.77 NTRK1 (0.44) NOS3NOS1NOS2
SCHEMBL13857012 0.73 SLC2A1 (0.55) SLC2A1KCNH2
SCHEMBL4270492 0.73 SLC2A1 (0.50) SLC2A1
SCHEMBL5797424 0.73 SLC2A1 (0.64) SLC2A1KCNH2
SCHEMBL14498889 0.68 KCNH2 (0.49) KCNH2
SCHEMBL4277304 0.68 GSK3A (0.42)
SCHEMBL14341258 0.67 KCNH2 (0.48) KCNH2
SCHEMBL14523985 0.67 KCNH2 (0.48) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7534793-B2 Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity SMITHKLINE BEECHAM P.L.C. (GB) 2009-05-19 US disclosed
US-7534793-B2 Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity SMITHKLINE BEECHAM P.L.C. (GB) 2009-05-19 US disclosed