SCHEMBL13859151

SCHEMBL13859151

CC(C)(F)[C@](C)(N)c1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 5/20 0.39
ACHE P22303 1/20 0.36
SLC22A12 Q96S37 2/20 0.35
KCNE1 P15382 1/20 0.35
KCNQ1 P51787 1/20 0.35
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HSD11B1 P28845 1/20 0.33
KIF11 P52732 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
ALDH1A1 P00352 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
POLB P06746 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30017695 0.79 KCNN4 (0.42) KCNN4ACHESLC22A12KCNE1KCNQ1
SCHEMBL1239429 0.79 KCNN4 (0.42) KCNN4ACHESLC22A12KCNE1KCNQ1
SCHEMBL3674130 0.79 KCNN4 (0.42) KCNN4ACHESLC22A12KCNE1KCNQ1
SCHEMBL12980626 0.79 KCNN4 (0.38) KCNN4SLC22A12KCNE1KCNQ1HDAC3
SCHEMBL14690376 0.79 KCNN4 (0.38) KCNN4SLC22A12KCNE1KCNQ1HDAC3
Hydrochloric Acid SCHEMBL26916930 0.77 KCNN4 (0.41) KCNN4ACHESLC22A12KCNE1KCNQ1
SCHEMBL2525080 0.77 KCNN4 (0.44) KCNN4ACHESLC22A12KCNE1KCNQ1
SCHEMBL20076543 0.77 ACHE (0.42) KCNN4ACHESLC22A12KCNE1KCNQ1
SCHEMBL11415516 0.77 ACHE (0.42) KCNN4ACHESLC22A12KCNE1KCNQ1
SCHEMBL15903165 0.76 KCNN4 (0.36) KCNN4KCNE1KCNQ1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2709992-A1 1,3-OXAZINES AS BACE1 AND/OR BACE2 INHIBITORS F. Hoffmann-La Roche AG (CH) 2014-03-26 EP disclosed
WO-2012156284-A1 1,3-OXAZINES AS BACE1 AND/OR BACE2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2012-11-22 WO disclosed