SCHEMBL13862136

SCHEMBL13862136

Nc1ccc(OCC(O)C(F)(F)F)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
CETP P11597 2/20 0.39
ALDH1A1 P00352 1/20 0.36
CFTR P13569 2/20 0.35
MGLL Q99685 1/20 0.35
ABHD6 Q9BV23 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
CYP1A2 P05177 1/20 0.34
MAOB P27338 1/20 0.34
AOC3 Q16853 1/20 0.34
PARP10 Q53GL7 2/20 0.33
PARP15 Q460N3 1/20 0.33
ADRB3 P13945 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8256645 0.81 MRGPRX4 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14301114 0.79 KMT2A (0.54) ALDH1A1MAOBAOC3ADRB3KMT2A
SCHEMBL6527647 0.78 APP (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL31552396 0.74 ALDH1A1 (0.48) ALDH1A1MAOBAOC3KMT2A
SCHEMBL31552390 0.74 ALDH1A1 (0.48) ALDH1A1HDAC1HDAC6MAOBAOC3
SCHEMBL27995830 0.74 MAOB (0.36) ALDH1A1HDAC1HDAC6CYP1A2MAOB
SCHEMBL27995828 0.74 MAOB (0.36) ALDH1A1HDAC1HDAC6CYP1A2MAOB
SCHEMBL9501793 0.73 ALDH1A1 (0.41) ALDH1A1HDAC1HDAC6
SCHEMBL13862109 0.73 ALDH1A1 (0.37) ALDH1A1MAOBPARP10ADRB3KMT2A
SCHEMBL9114780 0.73 MTNR1A (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622912-B1 2-ALKYNYL-AND 2-ALKENYL-PYRAZOLO- [4,3-E ] -1,2,4-TRIAZOLO- [1,5-C] -PYRIMIDINE ADENOSINE A2A RECEPTOR ANTAGONISTS SCHERING CORP (US) 2009-05-27 EP disclosed